一种5-取代的苯硫基-苯并咪唑-2-n-甲氧基羰基化合物的制备方法

Method for preparing 5-substituted thiophenyl-benzimidazol-2-N-methoxycarbonyl compound

Abstract

The invention discloses a method for preparing a 5-substituted thiophenyl-benzimidazol-2-N-methoxycarbonyl compound. In the method, a compound (I), a compound (II) and a compound (III) are synthesized respectively; and finally, a compound (IV) is synthesized. In the invention, the synthesis route is short, the raw material is cheap and readily available, the yield is high, the pollution is basically prevented, and industrial production can be carried out.
本发明一种5-取代的苯硫基-苯并咪唑-2-N-甲氧基羰基化合物的制备方法,本方法分别通过合成化合物(I)、化合物(II)、(III)最后合成化合物(IV)。本发明合成路线原料价格低廉易得、操作简单、收率高、污染小、适合工业化生产。

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Cited By (5)

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    CN-103073504-AMay 01, 2013湖南欧亚生物有限公司5-取代的苯硫基-苯并咪唑-2-n-甲氧基羰基氨基系列化合物的合成方法
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